Table 1

Taste and pheromone receptor gene (sub-)families in mice and Drosophila


Receptor
Number of intact genes
Conservation* within each family
Sites of expression
Known ligands (examples)
Structural notes

Mouse/ human
T1R
3 (human) 3 (mouse)
30-40%
Taste cells in the tongue; T1R1 plus T1R3 or T1R2 plus T1R3 are preferentially coexpressed, with few cells expressing all three genes
Sweet chemicals (T1R2 plus T1R3) L-amino acids, umami chemicals (T1R1 plus T1R3)
Similar to V2R (20-30% identical)

T2R
28 (human); approximately 40 (mouse)
25% to more than 80%
Taste cells in the tongue; most cells express many, if not all, T2R genes
Bitter compounds, such as cycloheximide (mouse T2R5), salicin (human T2R16), and PTC (human T2R38)
Similar to V1R (15-20% identical)

V1R
5 (human) 137 (mouse)
25% to nearly 100%
Basal layer in the vomeronasal organ; probably one V1R gene expressed per cell
2-heptanone (V1Rb1), 6-hydroxy-6-methyl-3-heptanone, n-pentylacetate, and isobutylamine
Similar to T2R (15-20% identical); important for maternal aggression

V2R
None in human; approximately 140 in mouse
25% to nearly 100%
Apical layer in the vomeronasal organ; probably one V2R gene expressed per cell
None identified
Similar to T1R (20-30% identical); forms a complex with MHC class Ib and β2-microglobulin; may be required for aggression between males

MHC 1b
None in human; 9 expressed in the mouse
40% to more than 80%
Apical layer in the vomeronasal organ; one or a few MHC 1b genes expressed per cell; coexpressed with a V2R gene
None (in the VNO)
Forms a complex with β2-microglobulin and V2Rs; may be required for aggression between males







Fly
GR
69
Approximately 15-75%
Spatially defined in one or several taste organs (labellum, labral and cibarial sense organs, legs, wings, and female genitalia)
Sugars and presumably other classes of compounds, including pheromones
Distantly related to olfactory receptor genes (Or83b); gustatory receptor probably recognize the whole spectrum of small soluble ligands; up to 20 subfamilies (with 1-8 genes each)

GR_S
8
44-75%
Foreleg and labellum (Gr5a), possibly other taste sensory organs
Trehalose (Gr5a)
The knockout fly has lower sensitivity to trehalose; member of a subfamily of 7 genes

*The numbers in this column refer to amino-acid sequence identity in mice and amino-acid sequence similarity in Drosophila, respectively. Indicates proposed rather than functionally established subfamilies of gustatory receptor genes that might function as sweet (S) receptors. This information is based on the functional characterization of a single receptor in this subfamily.

Matsunami and Amrein Genome Biology 2003 4:220   doi:10.1186/gb-2003-4-7-220